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新型糖氨基酸类化合物的合成研究
(2015)
Wang, Xuebin ; Wang, Xiaoli ; Hu, Jing ; Wang, Zhaoya ; Pimpalpalle, Tukaram M. ; Linker, Torsten ; Yin, Jian
Sugar amino acids (SAAs) are carbohydrate derivatives bearing both amino and carboxylic acid functional groups. SAAs represent an important class of multifunctional building blocks, which are amenable to serve as glycomimetics or peptidomimetics with well-defined structures and useful properties. Because SAAs exist in nature in many forms with various biological activities, recently, many unnatural SAAs, as the demand for finding new molecules to discover new drugs and new materials, have been designed and synthesized by a number of research groups. In this paper, we have developed a convenient method for the synthesis of novel SAAs gluco-7 and galacto-7 for the first time. The structure of gluco-7 was similar to the natural SAA glucosaminuronic acid that was a component of many typical bacterial cell walls and could be used for the preparation of type D flu vaccine; while galacto-7 was similar to the natural SAA galactosaminuronic acid that was one of bacterial Vi-antigen components of Escherichia coli. Starting from unexpensive and commercially available 3,4,6-tri-O-acetyl-D-glucal and 3,4,6-tri-O-acetyl-D-galactal, two novel SAAs gluco-7 and galacto-7 were achieved in the linear 6 steps with 34% overall yield and 19% overall yield, respectively. The key reactions included radical addition, decarboxylation, iodine generation reaction, azide reaction and reductive amination reaction. The crucial step was the synthesis of the target compound gluco-7 from gluco-6. By using method A, the target compound gluco-7 was obtained in 4 steps with 63% overall yield. To optimize the transformation from gluco-6 to gluco-7, method B was developed to generate gluco-7 by using one-pot reaction successfully with 76% yield only in one step. It proved that method B was superior to method A with shorter steps and higher yields. All the new compounds were characterized by IR, H-1 NMR, C-13 NMR and HRMS data. Study on the synthesis and biological evaluation of linear and cyclic oligomers derived from gluco-7 and galacto-7 are currently in progress.
Alexander von Humboldts 1827/28 gehaltene Kosmos-Vorträge stellen ebenso einen kanonischen Bezugspunkt wie einen weißen Fleck in der Rezeption seines Schaffens dar. Zahlreiche Deutungen basieren auf lediglich zwei unkommentierten Leseausgaben von Collegheften anonym gebliebener Zuhörer Humboldts. Seine 2009 wiedergefundenen eigenhändigen Vorlesungsmanuskripte versprechen, diese schmale Quellenbasis zu erweitern. Alfred Dove hatte bereits 1872 auf ihre Existenz verwiesen und interpretierte sie damals als Nukleus der schriftlichen Ausarbeitung des Kosmos. Diese Sichtweise hat sich in der Rezeption gehalten, während die Materialien, die Dove beschrieb, in Vergessenheit gerieten. Der Artikel stellt anhand ausgewählter Beispiele die Vorlesungsmanuskripte Humboldts und Nachschriften seiner Zuhörer in ihrem Zusammenhang vor, entwickelt die These von der Eigenständigkeit der sogenannten Kosmos-Vorträge gegenüber dem fünfbändigen Kosmos und umreißt die wichtigsten Ziele und Inhalte der geplanten digitalen Edition.
Die explorative hochschuldidaktische Studie geht der Frage nach, ob die Erfahrungen im Praxissemester und in den erziehungswissenschaftlichen Begleitseminaren dazu beitragen, die subjektive Sicht der Studierenden auf das erziehungswissenschaftliche Studium und den Nutzen einer erziehungswissenschaftlichen Reflexion eigener pädagogischer Praxis zu verändern. Die zentrale These des Beitrages lautet: Erst die reflektierte fallanalytische erziehungswissenschaftliche Auseinandersetzung mit der eigenen pädagogischen Praxis führt zu einer höheren Bedeutungszuschreibung an das erziehungswissenschaftliche Studium und lässt die Erziehungswissenschaft aus Sicht der Studierenden nach dem Praxissemester zur wichtigen Berufswissenschaft werden. Grundlage der Studie sind schriftliche Statements Studierender (n = 184) aus einem seminaristischen Reflexions- und Diskussionsprozess am Ende des Praxissemesters aus einem Zeitraum von acht Jahren. Abgeschlossen wurde der Beitrag im August 2019.
Gustav Rose (1798-1873) begleitete Alexander von Humboldt auf seiner Russlandreise und stand bis zu Humboldts Tod persönlich und postalisch zum ihm in Kontakt. Die Edition des vorliegenden Briefs zielt darauf ab, die Bedeutung der Person Gustav Rose in ihrer Beziehung zu Alexander von Humboldt und ihrem Einfluss auf den mineralogisch-geologischen Teil des Kosmos zu beleuchten und dem Leser dieses interessante historische Dokument zugänglich zu machen.
„The game’s afoot!“
(2020)
Computerspiele bieten – verstanden als Text, als popkulturelles Artefakt, als Lerngelegenheit und vieles mehr – auch für den Einsatz im Fremdsprachenunterricht zahlreiche Möglichkeiten, curricular vorgegebene Kompetenzen auszubilden. Nicht nur kann die Auseinandersetzung mit Computerspielen einen Beitrag zur fachintegrativen Vermittlung von Medienkompetenz leisten, sondern ebenso dazu genutzt werden, Handlungen zu simulieren, in denen Schülerinnen und Schüler fremdsprachig (inter-)agieren. Der folgende Beitrag versucht daher, exemplarisch zwei Computerspiele auf ihr Potential für den Einsatz im Fremdsprachenunterricht Englisch zu untersuchen. Er versteht sich als praktischer Beitrag, der Einblick in didaktisch-methodische Überlegungen bietet, welche die Auseinandersetzung mit den zwei exemplarisch ausgewählten Spielen, HER STORY (2015) und 1979 REVOLUTION: BLACK FRIDAY (2016), in den Blick nehmen.
Sprachbildung findet nicht nur im neuen Rahmenlehrplan für Berlin und Brandenburg explizit in allen Fächern Berücksichtigung, Sprachbildung ist gegenwärtig zugleich bundesweit eines der zentralen Themen der Lehrkräftebildung. In vorliegendem Beitrag werden zunächst Hintergründe sowie Ziele einer Verankerung von Sprachbildung in der Lehrkräftebildung präsentiert. Hieran anknüpfend werden die Grundzüge eines Konzepts für die Universität Potsdam präsentiert, an der Sprachbildung bislang noch nicht in den Studiengängen für das Lehramt für die Sekundarstufen verankert ist. Der Beitrag schließt mit Erfahrungen aus Lehrveranstaltungen zu Sprachbildung im Fach, die im Rahmen des Projekts „Sprachliche Heterogenität als Herausforderung in der Lehrkräftebildung“ gemacht wurden und in die zukünftige Entwicklung einfließen werden.
Der vorliegende Beitrag widmet sich einem Seminar in den Bildungswissenschaften, das im Rahmen von „PSI-Potsdam“ konzipiert wurde und seit dem Wintersemester 2016/17 jeweils einmal pro Semester umgesetzt wird. Die konzeptionelle Besonderheit der Lehrveranstaltung zeigt sich vor allem in der Zielgruppe: Das Seminar mit einem Umfang von 2 Semesterwochenstunden ist für Lehrer_innen als Fortbildungsveranstaltung geöffnet. Dadurch ergeben sich gemischte Seminargruppen, in denen die Teilnehmer_innen mit sehr unterschiedlichen Vorerfahrungen vertreten sind. Dennoch lassen sich Forschungs- und Praxisorientierung verbinden und darüber hinaus auch Impulse für die Schulpraxis setzen. Den Studierenden erweist sich die Seminarteilnahme zudem als Zugang zum (Forschungs-) Feld Schule.
Nicht nur der Lauf der Geschichte verändert sich, sondern auch Geschichtswissenschaft und -unterricht. An die Stelle des Auswendiglernens vorgegebener historischer Erzählungen trat im Laufe der Zeit zunehmend die Befähigung zu deren Dekonstruktion. Dafür müssen allerdings die Entstehungsbedingungen (geschichts-)wissenschaftlicher Erkenntnisse nachvollzogen werden können. Eine Möglichkeit, dies auf spielerische Art und Weise, aber auch auf Augenhöhe mit Lehrkräften und Historiker*innen zu tun, bieten Open-World- Spiele wie HORIZON ZERO DAWN (2017).